Bioactive Small Molecules
A vast array of small, non-peptide, organic compounds that are biologically active. Products include receptor antagonists, molecular probes, metabolites, GPCR ligands, neurotransmitters, ion channel modulators, and signaling activators and inhibitors.
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241
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241
Tocris Bioscience™ Nimbolide
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RNF114 inhibitor
| Target | Ubiquitin Ligase (E3) Inhibitors |
|---|---|
| CAS | 25990-37-8 |
| Purity | 0.97 |
| Chemical Name or Material | (2 aR,5 aR,6 S,6 aR,8 R,9 aR,10 AS,10 bR,10 cR)-8-(3-Furanyl)-2 A,5 A,6,6 A,8,9,9 A,10 A,10 b,10 c-decahydro-2 A,5 A,6 A,7-tetramethyl-2,5-dioxo-2 H,5 H-cyclopenta[d']naphtho[1,8-bc:2,3-b']difuran-6-acetic acid methyl ester |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C27H30O7 |
242
| CAS | 7770-78-7 |
|---|---|
| Molecular Formula | C21H24O6 |
243
Tocris Bioscience™ THPTA
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Click chemistry auxiliary reagent; accelerating ligand for copper-catalyzed azide-alkyne cycloaddition reaction
244
Tocris Bioscience™ DBCO-NHS
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Amine reactive and azide reactive building block
246
Tocris Bioscience™ FTBMT
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Potent and selective GPR52 agonist; orally bioavailable and BBB permeable
| CAS | 1358575-02-6 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 4-[3-[[3-Fluoro-5-(trifluoromethyl)phenyl]methyl]-5-methyl-1H-1,2,4-triazol-1-yl]-2-methylbenzamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H16F4N4O |
| Formula Weight | 392.35 |
247
Tocris Bioscience™ PZM21
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Selective μ receptor agonist
| Target | mu Opioid Receptor Agonists |
|---|---|
| CAS | 1997387-43-5 |
| Purity | 0.98 |
| Chemical Name or Material | N-[(2 S)-2-(Dimethylamino)-3-(4-hydroxyphenyl)propyl]-N'-[(1 S)-1-methyl-2-(3-thienyl)ethyl]urea |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C19H27N3O2S |
248
Tocris Bioscience™ MR 24
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective MST3 kinase binding inhibitor
| Target | Other Kinase Inhibitors |
|---|---|
| Purity | 0.98 |
| Chemical Name or Material | 8-(4-Aminobutyl)-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(1,3-dihydroxypropan-2-ylamino)pyrido[2,3-d]pyrimidin-7-one trihydrochloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C26H29ClN6O3.3HCl |
249
250
| CAS | 42017-89-0 |
|---|---|
| Molecular Formula | C17H15ClO4 |
251
| Target | Ferroptosis Inhibitors |
|---|---|
| CAS | 862808-01-3 |
| Purity | 0.98 |
| Chemical Name or Material | 3-(4-Bromophenyl)-6-((4-(4-methoxyphenyl)piperazin-1-yl)methyl)thiazolo[2,3-c][1,2,4]triazole |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C22H22BrN5OS |
252
| Target | Adrenergic alpha-2 Receptor Antagonists |
|---|---|
| CAS | 2313483-41-7 |
| Purity | 0.98 |
| Chemical Name or Material | 1-[2-[[[3-(3,5-Dimethyl-4-isoxazolyl)imidazo[1,2-a]pyridin-7-yl]carbonyl]amino]ethyl]-4-(methylamino)pyridinium chloride |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C21H23ClN6O2 |
253
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Tocris Bioscience™ NVS-STG2
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Tocris Bioscience™ NVS-STG2
Greener Choice
Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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STING agonist, molecular glue that causes oligomerization of STING
| Target | STING Agonists |
|---|---|
| CAS | 3030588-01-0 |
| Purity | 0.98 |
| Chemical Name or Material | 4-((4-(2-(tert-Butyl)-5,5-dimethyl-1,3-dioxan-2-yl)benzyl)amino)-3-methoxybenzoic acid |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C25H33NO5 |
254
| Shipping Condition | No special requirements |
|---|---|
| CAS | 58-46-8 |
| Color | White to Light-yellow to Beige |
| Purity | ≥97.5% |
| Physical Form | Crystalline Powder |
| Health Hazard 1 | Exclamation mark |
| Chemical Name or Material | Tetrabenazine |
| Recommended Storage | Refrigerator +4°C |
| Molecular Formula | C19 H27 N O3 |
| EINECS Number | 200-383-6 |
| Melting Point | 124°C to 130°C |
| Product Line | Life science |
255
Tocris Bioscience™ AZ 5704
Greener Choice
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Greener Choice
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Offers one or more environmental benefits itemized in the U.S. FTC “Green Guides.”
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Potent and selective ATM kinase inhibitor; orally bioavailable
| CAS | 1941214-06-7 |
|---|---|
| Purity | 98% |
| Chemical Name or Material | 7-Fluoro-6-[6-(methoxymethyl)-3-pyridinyl]-4-[[(1S)-1-(1-methyl-1H-pyrazol-3-yl)ethyl]amino]-3-quinolinecarboxamide |
| Recommended Storage | Store at -20°C |
| Molecular Formula | C23H23FN6O2 |
| Formula Weight | 434.47 |